PROGRAM · plogosertib (THT-140)

A next-generation oral PLK1 inhibitor.

Wholly owned by Tethra Biosciences; acquired in October 2025 from the Cyclacel chemistry estate. In active Phase 1/2 development across solid tumors and lymphoma; AML combination program planned for 2027.

Modality
Oral small molecule
Target
PLK1
Stage
Phase 1 / Phase 1/2
Origin
Cyclacel patent estate

Development across three tracks

Pipeline

Program
Indication
Stage
Status
Phase 1/2 trial · same protocol covers both indications Trial 1 · Active
Plogosertib PLK1 + BRD4 inhibitor · Tethra Bio
Solid tumors biomarker-defined
DiscoveryPreclin.INDPhase 1Phase 2
Active P1/2
Plogosertib PLK1-sensitive · Tethra Bio
Lymphoma biomarker-defined
DiscoveryPreclin.INDPhase 1Phase 2
Active P1/2
Plogosertib + Combination Combination · Tethra Bio
AML biomarker-defined
DiscoveryPreclin.INDPhase 1Phase 2
Planned 2027

Intellectual property

plogosertib's protection derives from the Cyclacel patent families, acquired by Tethra in October 2025. Coverage spans composition of matter and methods of use across major jurisdictions. A patent-status summary is available to qualified parties under CDA.

Regulatory

Tethra is pursuing standard FDA development pathways for plogosertib across its indication tracks. Designations, trial registrations, and protocol details will be disclosed through official regulatory channels.

Trials

Clinical trials

Trial listings coming soon

Active and planned trials will be linked here with ClinicalTrials.gov identifiers as records are updated.

Contact us
plogosertib (THT-140) is investigational and has not been approved by any health authority.